Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50145957'
TargetIntegrase(Human immunodeficiency virus 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145957((Z)-4-(3-{3-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of HIV-1 integrase catalytic activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3136PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Institute of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50145957((Z)-4-(3-{3-[3-(3-Carboxy-3-hydroxy-acryloyl)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Evaluated for inhibition of HIV-1 integrase catalytic activity in terms of inhibition of 3'-processingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P3136PubMed