Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Interstitial collagenase' and Ligand = 'BDBM50264809'
TargetInterstitial collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50264809(2-((4-phenoxyphenylsulfonyl)methyl)thiirane | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  7.30E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GB281XPubMed
TargetInterstitial collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50264809(2-((4-phenoxyphenylsulfonyl)methyl)thiirane | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  2.06E+5nMAssay Description:Competitive inhibition of human MMP1 using fluorogenic substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T43V4QPubMed
TargetInterstitial collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50264809(2-((4-phenoxyphenylsulfonyl)methyl)thiirane | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  2.06E+5nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD4WM2PubMed
TargetInterstitial collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50264809(2-((4-phenoxyphenylsulfonyl)methyl)thiirane | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  2.06E+5nMAssay Description:Inhibition of human recombinant MMP1 catalytic domain by substrate hydrolysis based fluorescence spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29X6GPubMed