Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50138766'
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50138766(CHEMBL439272 | cyclo[D-Ala3]Dyn A-(1-11)NH2)copy SMILEScopy InChI
Affinity DataKi:  0.210nMAssay Description:Binding affinity towards Opioid receptor kappa 1 expressed in CHO cells was determined by using [3H]-diprenorphine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q23ZN2PubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50138766(CHEMBL439272 | cyclo[D-Ala3]Dyn A-(1-11)NH2)copy SMILEScopy InChI
Affinity DataEC50:  0.540nMAssay Description:Inhibition of forskolin-stimulated adenylyl cyclase activity by compound in CHO cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q23ZN2PubMed