Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50580697'
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50580697(CHEMBL5071625)copy SMILES
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-diprenorphine from mouse KOR expressed in HEK293 cell membranes by radioligand binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0R4NPubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50580697(CHEMBL5071625)copy SMILES
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at EGFP-tagged mouse KOR expressed in HEK293 cells co-expressing beta-arrestin2 nano-luciferase assessed as beta-arrestin2 recruitme...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0R4NPubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))TBA
LigandPNGBDBM50580697(CHEMBL5071625)copy SMILES
Affinity DataEC50:  45nMAssay Description:Agonist activity at mouse KOR expressed in HEK293 cell assessed as inhibition of cAMP concentration incubated for 1 hrs by time-resolved fluorescence...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0R4NPubMed