Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50196462'
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50196462(CHEMBL3956072)copy SMILEScopy InChI
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000425PubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50196462(CHEMBL3956072)copy SMILEScopy InChI
Affinity DataEC50:  23nMAssay Description:Agonist activity at rat KISS1R expressed in CHO/dhfr cells assessed as increase in intracellular Ca2+ levels measured for 180 secs by Fluo 3-AM dye b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000425PubMed