Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50392411'
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M675SPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M675SPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP477RPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP477RPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of human KISS1R expressed in CHO cells assessed as inhibition of KISS1R-mediated cell growth after 4 days by cell counting kit-8 assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M675SPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50392411(CHEMBL2151652)copy SMILEScopy InChI
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP477RPubMed