Affinity DataKi: 0.120nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to human KISS1RMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human KISS1R expressed in CHO cells assessed as inhibition of KISS1R-mediated cell growth after 4 days by cell counting kit-8 assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.110nMAssay Description:Agonist activity at human KISS1R assessed as induction of intracellular calcium mobilization by fluorometric analysisMore data for this Ligand-Target Pair