Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50442964'
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50442964(CHEMBL3085809)copy SMILEScopy InChI
Affinity DataKi:  0.0440nMAssay Description:Binding affinity to human KISS1R expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M675SPubMed
TargetKiSS-1 receptor(Rattus norvegicus)
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50442964(CHEMBL3085809)copy SMILEScopy InChI
Affinity DataKi:  0.0590nMAssay Description:Binding affinity to rat KISS1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M675SPubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50442964(CHEMBL3085809)copy SMILEScopy InChI
Affinity DataEC50:  0.0570nMAssay Description:Agonist activity at human KISS1R expressed in CHO cells assessed as increase in calcium mobilization measured at 2 secs interval for 2 mins by fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD513CPubMed