Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Large neutral amino acids transporter small subunit 1' and Ligand = 'BDBM50174345'
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50174345(CHEMBL3809112)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Cis-inhibition of human LAT1 expressed in TREx HEK293 cells at 200 uM assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8J66PubMed
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50174345(CHEMBL3809112)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of human LAT1 expressed in HEK cells assessed as reduction in uptake of [3H]-gabapentin after 3 mins by scintillation counting based cis-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2ZFDPubMed