Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Large neutral amino acids transporter small subunit 1' and Ligand = 'BDBM50463186'
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University of Nebraska at Kearney

Curated by ChEMBL
LigandPNGBDBM50463186(CHEMBL4242404)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:Cis-inhibition of human LAT1 expressed in TREx HEK293 cells assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 degC follo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JBJPubMed
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
University of Nebraska at Kearney

Curated by ChEMBL
LigandPNGBDBM50463186(CHEMBL4242404)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:Cis-inhibition of human LAT1 expressed in TREx HEK293 cells at 200 uM assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8J66PubMed