Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Lethal(3)malignant brain tumor-like protein 3' and Ligand = 'BDBM50440603'
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50440603(CHEMBL2426498)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50440603(CHEMBL2426498)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50440603(CHEMBL2426498)copy SMILEScopy InChI
Affinity DataKd:  390nMAssay Description:Binding affinity to L3MBTL3 (unknown origin) by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27WRPPubMed