Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4E' and Ligand = 'BDBM19149'
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of JMJD2E pre-incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X870SPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W95F76PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 5.40E+5nMpH: 7.5 T: 2°CAssay Description:A coupled-assay for JMJD2E activity employing formaldehyde dehydrogenase (FDH) from Pseudomonas putida was developed. Formaldehyde release by demethy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959FV4PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 5.40E+5nMAssay Description:Inhibition of JMJD2EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X870SPubMed