Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4E' and Ligand = 'BDBM50396018'
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human N-terminal His6-tagged KDM4E catalytic domain (1 to 337 residues) expressed in Escherichia coli using ARK(me3)STGGK as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP5559PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8X83PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant JMJD2E (unknown origin) incubated for 15 mins prior to substrate addition by AlphaScreen methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028VHDPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of KDM4E (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0RBNPubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human N-terminal His6-tagged KDM4E catalytic domain (1 to 337 residues) expressed in Escherichia coli using ARK(me3)STGGK as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP5559PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50396018(CHEMBL1230640)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of JMJD2E catalytic domain by mass spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ62NXPubMed