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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 5A/5B' and Ligand = 'BDBM264001'
Target
Lysine-specific demethylase 5A/5B
(Homo sapiens (Human))
Celgene Corporation
Curated by
ChEMBL
Ligand
BDBM264001
(2-{5-[(4-chloro-2- fluorobenzyl)oxy]-1H-pyrazol-1-...)
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Affinity Data
EC50: 1.30E+3nM
Assay Description:
Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26Q20W4
PubMed