Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Lysophosphatidic acid receptor 2' and Ligand = 'BDBM50148348'
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)copy SMILEScopy InChI
Affinity DataEC50:  6.80nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50MDWPubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)copy SMILEScopy InChI
Affinity DataEC50:  29nMAssay Description:Agonist activity at human LPA2 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HS4PubMed