Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'MAP kinase-activated protein kinase 2' and Ligand = 'BDBM50395275'
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma Ltd.

Curated by ChEMBL
LigandPNGBDBM50395275(CHEMBL2163616)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K29PXPubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma Ltd.

Curated by ChEMBL
LigandPNGBDBM50395275(CHEMBL2163616)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human MAPKAP-K2 in THP1 cells assessed as inhibition of LPS-induced TNFalpha production incubated 1 hr prior to LPS challenge measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K29PXPubMed