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TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma Ltd.
Curated by ChEMBL
Teijin Pharma Ltd.
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of MAPKAP-K2 using KKLNRTLSVA as substrate and [33P]-gamma-ATP after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Teijin Pharma Ltd.
Curated by ChEMBL
Teijin Pharma Ltd.
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human MAPKAP-K2 in THP1 cells assessed as inhibition of LPS-induced TNFalpha production incubated 1 hr prior to LPS challenge measured ...More data for this Ligand-Target Pair
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