Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'MAP kinase-interacting serine/threonine-protein kinase 1' and Ligand = 'BDBM50455558'
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)

Curated by ChEMBL
LigandPNGBDBM50455558(CHEMBL4213023)copy SMILEScopy InChI
Affinity DataIC50: 528nMAssay Description:Inhibition of GST-tagged MNK1 (37 to 341 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) using JH3 peptide as substrate preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20004P7PubMed