Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM50363397'
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Concentration required to inhibit the activity of K+ stimulated gastric ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4FN0PubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3WQ4PubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
TU Dortmund University

Curated by ChEMBL
LigandPNGBDBM50363397(CHEMBL1946170 | REGORAFENIB | US10183928, Regorafe...)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Inhibition of recombinant N-terminal 6x-His-tagged c-KIT (547 to 935 residues)/(694 to 753 residues deletion) (unknown origin) expressed in baculovir...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7M1WPubMed