Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50197139'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MCH from MCHr1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4Q7PPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of 125I-MCH from MCH-R1 expressed in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50MMKPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29WNWPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity at MCHR1 assessed as inhibition of MCH-mediated calcium release in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29WNWPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197139(CHEMBL214021 | N-(1-(benzo[d][1,3]dioxol-5-ylmethy...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity at MCHr1 assessed as inhibition of MCH-mediated calcium ion release in intact IMR32 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4Q7PPubMed