Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50207681'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207681(CHEMBL248297 | N-(1-(3-fluoro-4-(3-(piperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MCH from MCHR1 expressed in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29WNWPubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50207681(CHEMBL248297 | N-(1-(3-fluoro-4-(3-(piperidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Antagonist activity at MCHR1 assessed as inhibition of MCH-mediated calcium release in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29WNWPubMed