Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50219041'
Affinity DataKi: 14nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at rat MCHR1 expressed in HEK293 cells assessed as effect on calcium mobilizationMore data for this Ligand-Target Pair