Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 3' and Ligand = 'BDBM50581319'
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50581319(BIM-22493 | RM-493 | SETMELANOTIDE | Setmelanotide)copy SMILES
Affinity DataKi:  13nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK2936E cell membrane measured after 16-23 hrs by 1450 microbeta trilux scintillat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50581319(BIM-22493 | RM-493 | SETMELANOTIDE | Setmelanotide)copy SMILES
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50R5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50581319(BIM-22493 | RM-493 | SETMELANOTIDE | Setmelanotide)copy SMILES
Affinity DataEC50:  0.151nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50R5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50581319(BIM-22493 | RM-493 | SETMELANOTIDE | Setmelanotide)copy SMILES
Affinity DataEC50:  0.151nMAssay Description:Agonist activity at human melanocortin receptor 3 expressed in human T-REx-293 cells assessed as stimulation of intracellular cAMP accumulation incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed