Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50340463'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340463(CHEMBL1761871 | cis-(3S,5R)-N-((R)-1-(4-(tert-buty...)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3S0GPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340463(CHEMBL1761871 | cis-(3S,5R)-N-((R)-1-(4-(tert-buty...)copy SMILEScopy InChI
Affinity DataEC50:  13nMAssay Description:Agonist activity at human MC4 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3S0GPubMed