Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50453132'
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)copy SMILEScopy InChI
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed