Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50581318'
TargetMelanocortin receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50581318(CHEMBL5076315)copy SMILES
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK2936E cell membrane measured after 16-23 hrs by 1450 microbeta trilux scintillat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50581318(CHEMBL5076315)copy SMILES
Affinity DataEC50:  1nMAssay Description:Agonist activity at human melanocortin receptor 4 expressed in human T-REx-293 cells using high doxycycline assessed as stimulation of intracellular ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50581318(CHEMBL5076315)copy SMILES
Affinity DataEC50:  32nMAssay Description:Agonist activity at human melanocortin receptor 4 expressed in human T-REx-293 cells using low doxycycline assessed as stimulation of intracellular c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301TQPubMed