Found 13 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM50121900'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
H. Lee Moffitt Cancer Center& Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center& Research Institute
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0380nMAssay Description:Activity in mouse melanocortin-1 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0380nMAssay Description:In vitro activaction of mouse recombinant Melanocortin-1 receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 0.0380nMAssay Description:Agonist activity to the mouse Melanocortin-1 receptor (mMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.380nMAssay Description:Effective concentration against mouse Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0880nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0320nMAssay Description:In vitro agonist potency for Mouse Melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0230nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0500nMAssay Description:Agonist activity at mouse MC1 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0140nMAssay Description:Agonistic activity against mouse MC1RMore data for this Ligand-Target Pair
Affinity DataEC50: 0.00800nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0300nMAssay Description:Functional activity at the mouse melanocortin 1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0180nMAssay Description:Effective concentration for mouse Melanocortin-1 receptorMore data for this Ligand-Target Pair