Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1C' and Ligand = 'BDBM85065'
TargetMelatonin receptor type 1C(Gallus gallus)
University College London

Curated by ChEMBL
LigandPNGBDBM85065(CAS_117946-91-5 | Luzindole | NSC_122162)copy SMILEScopy InChI
Affinity DataKi:  1.61E+3nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154KSHPubMed
TargetMelatonin receptor type 1C(Xenopus)
King's College London

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | Luzindole | NSC_122162)copy SMILEScopy InChI
Affinity DataKi:  2.04E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7G6SPubMed
TargetMelatonin receptor type 1C(Xenopus)
King's College London

Curated by PDSP Ki Database
LigandPNGBDBM85065(CAS_117946-91-5 | Luzindole | NSC_122162)copy SMILEScopy InChI
Affinity DataIC50: 2.46E+3nMAssay Description:Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859BKPubMed