Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50105833'
TargetMetabotropic glutamate receptor 1(RAT)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0HX0PubMed
TargetMetabotropic glutamate receptor 1(RAT)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)copy SMILEScopy InChI
Affinity DataIC50: 207nMAssay Description:Negative allosteric modulatory activity at rat cloned mGluR1 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced calci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0HX0PubMed