Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50252048'
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at rat mGluR1 expressed in HEK293 cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu1 receptor expressed in HEK293 cells by intracellular Ca2+ mobilization assayMore data for this Ligand-Target Pair