Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 2' and Ligand = 'BDBM50034504'
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataKi:  300nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M043ZHPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M61HS5PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataKi:  490nMAssay Description:Agonist potency against cloned Metabotropic glutamate receptor 2 agonistMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DZ090QPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataEC50:  750nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR2 in ratMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20R9Q1RPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataEC50:  380nMAssay Description:Concentration for half maximal activation of metabotropic glutamate mGluR2 in humanMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20R9Q1RPubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Emory University

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat nonneuronal cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K936Z5PubMed