Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50139452'
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50139452(CHEMBL3764943)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]MPEP from rat mGlu5 receptor expressed in rat cerebrocortical membrane measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930W1NPubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50139452(CHEMBL3764943)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]M-MPEP from mGluR5 in Sprague-Dawley rat cerebrocortical membranes after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R05PubMed
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Gedeon Richter Plc

Curated by ChEMBL
LigandPNGBDBM50139452(CHEMBL3764943)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]M-MPEP from recombinant human mGluR5a expressed in human A18 cell membrane homogenate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R05PubMed