Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50252051'
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at rat mGluR5 expressed in HEK293 cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Universite Blaise Pascal
Curated by ChEMBL
Universite Blaise Pascal
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu5 receptor expressed in HEK293 cells by intracellular Ca2+ mobilization assayMore data for this Ligand-Target Pair