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Affinity DataKi: 17nMAssay Description:Displacement of [3H]-MPEP from mGluR5 in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Modulation of human recombinant mGluR5 expressed in CHO cells assessed as inhibition of glutamate-induced responseMore data for this Ligand-Target Pair
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