Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 5' and Ligand = 'BDBM50429420' TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 760nMAssay Description:Displacement of [3H]-ABP688 from human mGluR5 expressed in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Antagonist activity at human mGluR5 expressed in HEK293 cells assessed as inhibition of Ca2+ mobilization by FLIPR assayMore data for this Ligand-Target Pair
