Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM120127'
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.

US Patent
LigandPNGBDBM120127(US8697715, Beta | US9259470, Beta)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4NSQUS Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Array BioPharma Inc.; Genentech, Inc.

US Patent
LigandPNGBDBM120127(US8697715, Beta | US9259470, Beta)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9GXFUS Patent