Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM50248938'
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM

US Patent
LigandPNGBDBM50248938(CHEMBL4089284 | US10981896, Compound 21)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Candidates for inhibitor selectivity characterization were chosen based on an initial single-timepoint commercial kinome profiling screen performed w...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24X5BWVUS Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM

US Patent
LigandPNGBDBM50248938(CHEMBL4089284 | US10981896, Compound 21)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of ERK2 (unknown origin) using Ets-1 as substrate measured after 30 mins in presence of [gamma32P]ATP by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833VFFPubMed