Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 10' and Ligand = 'BDBM50234890'
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen

Curated by ChEMBL
LigandPNGBDBM50234890(CHEMBL4077018)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant 6x-His-tagged JNK3 (39 to 402 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2891854PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen

Curated by ChEMBL
LigandPNGBDBM50234890(CHEMBL4077018)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity against beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
In DepthDetails
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen

Curated by ChEMBL
LigandPNGBDBM50234890(CHEMBL4077018)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4NSBPubMed