Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12' and Ligand = 'BDBM50059253'
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Amgen

LigandPNGBDBM50059253(CHEMBL3393311 | US9868720, No. 3)copy SMILEScopy InChI
Affinity DataKi:  691nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38VWNUS Patent
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Amgen

LigandPNGBDBM50059253(CHEMBL3393311 | US9868720, No. 3)copy SMILEScopy InChI
Affinity DataKi:  691nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DJ5PubMed