Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12' and Ligand = 'BDBM50128338' TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
WuXi AppTec Co., Ltd.
Curated by ChEMBL
WuXi AppTec Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of N-terminally GST- tagged human DLK catalytic domain (1 to 520 amino acids) using N-terminally HIS-tagged MKK4 K131M as substrate incuba...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
WuXi AppTec Co., Ltd.
Curated by ChEMBL
WuXi AppTec Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 632nMAssay Description:Inhibition of Dox inducible human DLK transfected in HEK293 cells assessed as reduction in JNK phosphorylation incubated for 5.5 hrs measured by Hoec...More data for this Ligand-Target Pair
