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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Mitotic checkpoint serine/threonine-protein kinase BUB1' and Ligand = 'BDBM367339'
Target
Mitotic checkpoint serine/threonine-protein kinase BUB1
(Homo sapiens (Human))
Pfizer
Ligand
BDBM367339
((6RS)-6-(Hydroxymethyl)-6-methyl-3-(phenylamino)-2...)
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Affinity Data
IC50: 8nM
Assay Description:
Bub1-inhibitory activities of compounds described in the present invention were quantified using a time-resolved fluorescence energy transfer (TR-FRE...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2QN6931
US Patent