Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM438853'
TargetMu-type opioid receptor(Homo sapiens (Human))
Alkermes, Inc.

US Patent
LigandPNGBDBM438853(3-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Membrane protein from CHO (Chinese Hamster Ovarian) cells that stably expressed one type of the cloned human opioid receptor were incubated with 12 d...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RN3BWXUS Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Alkermes, Inc.

US Patent
LigandPNGBDBM438853(3-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0J91US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Alkermes, Inc.

US Patent
LigandPNGBDBM438853(3-((1R,5S,9R)-3-((1R,3r,5S)-6,6-difluorobicyclo[3....)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:The Ki (binding affinity) for μ-receptor was determined with a previously described method using a competitive displacement assay (Neumeyer et a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24J0J91US Patent