Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50139011'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  47.7nMAssay Description:Displacement of [3H]-endomorphin-2 from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  104nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  104nMAssay Description:Displacement of [3H]-DAMGO from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  107nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataIC50: 589nMAssay Description:Inhibition of Opioid receptor mu 1 of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(MOUSE)
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139011((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Mu opioid receptor of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed