Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50182942'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Binding affinity to rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DP8PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5MDZPubMed
TargetMu-type opioid receptor(GUINEA PIG)
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)copy SMILEScopy InChI
Affinity DataEC50:  27nMAssay Description:Activity against mu opioid receptor by stimulation of [35S]GTPgammaS binding in CHO-hgamma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5MDZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Janssen Research and Development, L.L.C.

Curated by ChEMBL
LigandPNGBDBM50182942((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-((S...)copy SMILEScopy InChI
Affinity DataEC50:  27nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DP8PubMed