Compile Data Set for Download or QSAR
Found 8 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50191056'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.970nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30Z0PubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Activity at mu opioid receptor by GPI/LMMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B30Z0PubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of mu opioid receptor in guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of electrically-stimulated musc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of mu opioid receptor in guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of electrically-stimulated musc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataEC50:  60nMAssay Description:Agonist activity at rat mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191056((S)-2-amino-3-(4-hydroxy-phenyl)-N-((R)-1-{[((S)-1...)copy SMILEScopy InChI
Affinity DataEC50:  69nMAssay Description:Agonist activity at rat mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T72MCMPubMed