Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50238615'
TargetMu-type opioid receptor(Homo sapiens (Human))
The University of Iowa

Curated by ChEMBL
LigandPNGBDBM50238615(CHEMBL264967 | Thiophene-2-carboxylic Acid (2S,4aR...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KR7PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The University of Iowa

Curated by ChEMBL
LigandPNGBDBM50238615(CHEMBL264967 | Thiophene-2-carboxylic Acid (2S,4aR...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [125]OXY from mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3D22PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The University of Iowa

Curated by ChEMBL
LigandPNGBDBM50238615(CHEMBL264967 | Thiophene-2-carboxylic Acid (2S,4aR...)copy SMILEScopy InChI
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human recombinant mu opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1KR7PubMed