Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50352115'
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)copy SMILEScopy InChI
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9B57PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)copy SMILEScopy InChI
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]Naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32SKPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9B57PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50352115(CHEMBL1824510 | CHEMBL1852385)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTP-gammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32SKPubMed