Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50558603'
TargetMu-type opioid receptor(MOUSE)TBA
LigandPNGBDBM50558603(CHEMBL4761986)copy SMILES
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]NLX from mouse MOR expressed in CHO cell membrane incubated for 90 mins by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD80CCPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50558603(CHEMBL4761986)copy SMILES
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human MOR transfected in CHO cells co-transfected with Gqi5 assessed as inhibition of DAMGO-induced calcium mobilization incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD80CCPubMed