Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50139772'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Queen's University

Curated by ChEMBL
LigandPNGBDBM50139772(22-oxovincaleukoblastine | leurocristine | vincris...)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.05 uM) in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PC33NHPubMed