Found 25 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50018056'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(GUINEA PIG)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 52nMAssay Description:Compound was evaluated for displacement of [3H]-QNB from human Muscarinic m2 receptor in CHO cells.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataKi: 81nMAssay Description:Binding affinity to human M2 muscarinic receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataIC50: 50nMAssay Description:Inhibition of muscarinic (M2) receptor isolated from rat atriaMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataIC50: 140nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataIC50: 400nMAssay Description:Inhibition of muscarinic (M2) receptor isolated from rat atriaMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataIC50: 400nMAssay Description:Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Université Louis Pasteur-Strasbourg
Curated by PDSP Ki Database
Affinity DataIC50: 400nMAssay Description:Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]-N-methylscopolamine as radioligandMore data for this Ligand-Target Pair