Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50265998'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265998(CHEMBL4070155)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]UNSW-MK259 from human muscarinic acetylcholine receptor M2 expressed in CHOK9 cells after 3 hrs by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1THCPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265998(CHEMBL4070155)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-NMS from human muscarinic M2 receptor expressed in CHO-K9 cells measured after 60 mins by Hoechst H33342 dye based confocal plat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R214WTPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265998(CHEMBL4070155)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Displacement of 4-(2-((1E,3E)-5-((E)-3,3-Dimethyl-1-(6-oxo-6-((2-(4-(4-(1-(2-oxo-2-(11-oxo-10,11-dihydro-5H-dibenzo[b,e][1,4]diazepin-5-yl)ethyl)pipe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R214WTPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265998(CHEMBL4070155)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]NMS from human muscarinic acetylcholine receptor M2 expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1THCPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50265998(CHEMBL4070155)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]UR-AP060 from human muscarinic acetylcholine receptor M2 expressed in CHOK9 cell homogenate after 3 hrs by liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1THCPubMed