Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50291551'
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a con...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RZ2
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.74E+4nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RZ2